Setmelanotide TFA
CAS No.
Setmelanotide TFA ( RM-493 TFA; BIM-22493 TFA; IRC-022493 TFA )
Catalog No. M29740 CAS No.
Setmelanotide TFA (RM-493 TFA; BIM-22493 TFA; IRC-022493 TFA) is a selective melanocortin 4 receptor (MC4R) agonist.
Setmelanotide TFA (RM-493 TFA; BIM-22493 TFA; IRC-022493 TFA) is a selective melanocortin 4 receptor (MC4R) agonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameSetmelanotide TFA
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NoteResearch use only, not for human use.
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Brief DescriptionSetmelanotide TFA (RM-493 TFA; BIM-22493 TFA; IRC-022493 TFA) is a selective melanocortin 4 receptor (MC4R) agonist.
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DescriptionSetmelanotide TFA (RM-493 TFA; BIM-22493 TFA; IRC-022493 TFA) is a selective melanocortin 4 receptor (MC4R) agonist.
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In Vitro
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In Vivo
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SynonymsRM-493 TFA; BIM-22493 TFA; IRC-022493 TFA
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PathwayOthers
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TargetOther Targets
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RecptorEC50: 5.8 nM (hMC1R), 5.3 nM (hMC3R), 0.27 nM (hMC4R), 0.28 nM (rMC4R), 1600 nM (hMC5R)
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Research Area
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Indication
Chemical Information
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CAS Number--
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Formula Weight1231.33
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Molecular FormulaC51H69F3N18O11S2
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Purity>98% (HPLC)
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Solubility
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SMILES
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Chemical Name
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
Kumar KG, et al. Analysis of the therapeutic functions of novel melanocortin receptor agonists in MC3R- and MC4R-deficient C57BL/6J mice. Peptides. 2009 Oct;30(10):1892-900.
molnova catalog
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